Palladium-catalyzed direct arylation of indoles with arylsulfonyl hydrazides.
نویسندگان
چکیده
A novel method to synthesise 2-arylindoles is demonstrated via direct arylation of indoles with arylsulfonyl hydrazides. Under the optimized reaction conditions, the reaction well tolerates a wide variety of functional groups to afford structurally diverse 2-arylindoles in good to excellent yields at 70 °C.
منابع مشابه
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عنوان ژورنال:
- Organic & biomolecular chemistry
دوره 14 10 شماره
صفحات -
تاریخ انتشار 2016